Wei Wang

KMap

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As Co-Director of the Arizona Center for Drug Discovery and professor in the Department of Pharmacology and Toxicology, Dr. Wang is responsible for advancing the mission of drug discovery at the UA Health Sciences, main campus and the Phoenix Biomedical Campus. By uniting the UA’s state-of-the-art facilities, expertise and resources, he will help facilitate drug discovery and development while enhancing translational research collaboration.

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Courses

IPDDP
Introduction to Pharmacology, Drug Discovery & Pharmaceutics
IMTDD
Introduction to Molecular Therapeutics and Drug Discovery
PDDDD
Principles in Drug Discovery, Design, and Development

MC
Medicinal Chemistry

Grants

Development of Inhibitors Targeting Flavivirus Methyltransferase
Co-Investigator (COI)
2023
$767.4K
Active
Novel Combinations of Natural Product Compounds for Treatment of Alzheimer Disease and Related Dementias
Principal Investigator (PI)
2023
$275.7K
Active
Novel Therapeutics for Pulmonary Hypertension
Co-Investigator (COI)
2022
$2.6M
Active
Discovery of PROTAC degraders of the SARS-Cov-2 main protease for the treatment of Covid-19
Co-Investigator (COI)
2022
$50.0K
Active
PTPRD Phosphatase Inhibitors for Stimulant Use Disorders
Principal Investigator (PI)
2022
$38.4K
Active
MRI: Acquisition of a Single-Crystal X-Ray Diffractometer for Research and Education
Co-Investigator (COI)
2021
$266.2K
Active
Discovery of PDE2A Inhibitors to Treat Memory Deficits in Mild Cognitive Impairment And Alzheimer's Disease
Principal Investigator (PI)
2021
$75.0K
Active
Design of Fe2+ and H2O2 Induced Proximity Functionalized Imaging Probes for the Control of Cellular Functions
Principal Investigator (PI)
2019
$1.3M
Active
Organocatalytic Practical Synthesis of Deuterated Building Blocks and Biologically Important Structures
Principal Investigator (PI)
2018
$1.1M
Active

PTPRD Ligands for Stimulant and Opiate Use Disorders
Principal Investigator (PI)
2019
$809.1K

News

UArizona Researchers Pivot to Tackle COVID-19
2020

Publications (371)

Recent

Organophotocatalytic silyl transfer of silylboranes enabled by methanol association: a versatile strategy for C–Si bond construction
2023
Controlling antifungal activity with light: Optical regulation of fungal ergosterol biosynthetic pathway with photo-responsive CYP51 inhibitors
2023
Site-selective deuteration at the α-position of enals by an amine and bis (phenylsulfonyl) methane co-catalyzed H/D exchange reaction
2022
Building bioorthogonal click-release capable artificial receptors on cancer cell surface for imaging, drug targeting and delivery
2022
A PET-based fluorescent probe for monitoring labile Fe (ii) pools in macrophage activations and ferroptosis
2022
Selective skeletal editing of polycyclic arenes using organophotoredox dearomative functionalization
2022
Synthesis of 2-oxoquinoline derivatives as dual pim and mTORC protein kinase inhibitors
2022
Methylglyoxal produced by tumor cells through formaldehyde-enhanced Warburg effect potentiated polarization of tumor-associated macrophages
2022
Orlistat increases arsenite tolerance in THP-1 derived macrophages through the up-regulation of ABCA1
2022
An anthracenecarboximide-guanidine fluorescent probe for selective detection of glyoxals under weak acidic conditions
2022
Structure-activity studies of PTPRD phosphatase inhibitors identify a 7-cyclopentymethoxy illudalic acid analog candidate for development
2022
Synthesis of C-1 Deuterated 3-Formylindoles by Organophotoredox Catalyzed Direct Formylation of Indoles with Deuterated Glyoxylic Acid
2022
Designing Efficient Cascade Reactions in Drug Discovery
2022
Synthesis of α-Aryl Primary Amides from α-Silyl Nitriles and Aryl Sulfoxides through [3, 3]-Sigmatropic Rearrangement
2022
Design of Photoredox-Catalyzed Giese-Type Reaction for the Synthesis of Chiral Quaternary α-Aryl Amino Acid Derivatives via Clayden Rearrangement
2022
Organophotocatalyzed E and Z stereoselective Csp3-Csp2 bond forming cross coupling reactions of carboxylic acids with β-aryl-vinyl halides
2021
Compositions and methods for controlling cellular function
2021
Photoredox Asymmetric Nucleophilic Dearomatization of Indoles with Neutral Radicals
2021
Construction of Enantioenriched γ, γ-Disubstituted Butenolides Enabled by Chiral Amine and Lewis Acid Cascade Cocatalysis
2021
Homo-PROTAC mediated suicide of MDM2 to treat non-small cell lung cancer
2021
A compact fluorescence/circular dichroism dual-modality probe for detection, differentiation, and detoxification of multiple heavy metal ions via bond-cleavage cascade reactions
2021
Synthesis of β-Silyl α-Amino Acids via Visible-Light-Mediated Hydrosilylation
2021
Aminocatalytic stereoselective synthesis of (E)-α-naphthyl enals via cross-coupling-like reaction of 1-bromo-2-naphthols with enals
2021
Formaldehyde reinforces pro-inflammatory responses of macrophages through induction of glycolysis
2021
Facile Synthesis of 2H-Benzo [h] Chromenes via an Arylamine-Catalyzed Mannich Cyclization Cascade Reaction
2021
Organophotocatalytic dearomatization of indoles, pyrroles and benzo (thio) furans via a Giese-type transformation
2021
PIFA‐Mediated Cross‐Dehydrogenative Coupling of N‐Heteroarenes with Cyclic Ethers: Ethanol as an Efficient Promoter
2021
An “AND”-logic-gate-based fluorescent probe with dual reactive sites for monitoring extracellular methylglyoxal level changes of activated macrophages
2021
Fluorophore-Promoted Facile Deprotonation and Exocyclic Five-Membered Ring Cyclization for Selective and Dynamic Tracking of Labile Glyoxals
2020
Copper Promoted Aerobic Oxidative C(sp3)–C(sp3) Bond Cleavage of N-(2-(Pyridin-2-yl)-ethyl)anilines
2020
Fluorescent Detection of Dynamic H2O2/H2S Redox Event in Living Cells and Organisms
2020
Graphitic Carbon Nitride Polymer as a Recyclable Photoredox Catalyst for Decarboxylative Alkynylation of Carboxylic Acids
2020
Catalytic asymmetric Catellani-type reaction: A powerful tool for axial chirality construction
2020
Organophotoredox-Catalyzed Formation of Alkyl–Aryl and− Alkyl C–S/Se Bonds from Coupling of Redox-Active Esters with Thio/Selenosulfonates
2020
Direct, stereoselective thioglycosylation enabled by an organophotoredox radical strategy
2020
Enantioselective [4+ 2] Cycloaddition Reaction of Vinylquinolines with Dienals Enabled by Synergistic Organocatalysis
2020
Deuteration of Formyl Groups via a Catalytic Radical H/D Exchange Approach
2020
An allosteric modulator of RNA binding targeting the N-terminal domain of TDP-43 yields neuroprotective properties
2020
Aldehydes Switch Regioselectivity: a Prins Cyclization Strategy for the Synthesis of Indoline‐fused THFs and Indole‐fused Oxepanes
2020
Mebendazole is a potent inhibitor to chemoresistant T cell acute lymphoblastic leukemia cells
2020
Potent Dual BET/HDAC Inhibitors for Efficient Treatment of Pancreatic Cancer
2020
One-pot synthesis of salicylaldehyde containing biaryl frameworks via an aminocatalytic Diels-Alder-retro-Diels-Alder cascade reaction of ynals with 2-pyrones
2020
Investigation of the Relationship Between H2O2 and HClO in Living Cells by a Bifunctional, Dual-ratiometric Responsive Fluorescent Probe
2020
Synthesis of Enantioenriched α-Deuterated α-Amino Acids Enabled by an Organophotocatalytic Radical Approach
2020
Autophagy: New Insights into Its Roles in Cancer Progression and Drug Resistance
2020
Visible light-mediated radical process for the synthesis of C-glycoamino acids
2019
Construction of N-Alkyl- and N-Arylaziridines from Unprotected Amines via C–H Oxidative Amination Strategy
2019
Organocatalytic thioesterification of aldehydes with visible light
2019
Trideuteromethylation Enabled by a Sulfoxonium Metathesis Reaction
2019
Moving beyond hydroxychloroquine: the novel lysosomal autophagy inhibitor ROC-325 shows significant potential in preclinical studies
2019
The Employment of Sodium Hydride as a Michael Donor in Palladium‐catalyzed Reductions of α, β‐Unsaturated Carbonyl Compounds
2019
Organocatalytic transformation of aldehydes to thioesters with visible light
2019
Photocatalytic C–H silylation of heteroarenes by using trialkylhydrosilanes
2019
Practical synthesis of C1 deuterated aldehydes enabled by NHC catalysis
2019
Highly stereoselective synthesis of aryl/heteroaryl-C-nucleosides via the merger of photoredox and nickel catalysis
2019
Fluorescence imaging of Fe (II) flux in ischemic stroke
2019
Synthesis of 3-aminoindan-1-one derivatives from 2-acetylbenzaldehydes and secondary amines by Mannich annulation
2019
A naphthalimide-aminal-based pH-sensitive fluorescent donor for lysosome-targeted formaldehyde release and fluorescence turn-on readout
2019
Visible-Light-Mediated, Chemo- and Stereoselective Radical Process for the Synthesis of C-Glycoamino Acids
2019
Improving the potency of cancer immunotherapy by dual targeting of IDO1 and DNA
2018
A Simple Two-photon Turn-on Fluorescent Probe for Selective Detection of Cysteine Based on Dual PeT/ICT Mechanism
2018
Monomethylarsonous Acid: Induction of DNA Damage and Oxidative Stress in Mouse Natural Killer Cells at Environmentally-relevant Concentrations
2018
α-Functionalization of 2-vinylpyridines via a chiral phosphine catalyzed enantioselective cross Rauhut–Currier reaction
2018
A simple two-photon turn-on fluorescent probe for the selective detection of cysteine based on a dual PeT/ICT mechanism
2018
Role of an isoform-specific residue at the calmodulin-heme (NO synthase) interface in the FMN - heme electron transfer
2018
Facile Synthesis of 2-Quinolinones via Hypervalent Iodine(III)-Mediated Intramolecular Decarboxylative-Heck Reaction at Room Temperature
2018
Organocatalytic Asymmetric Formal [4 + 2] Cycloaddition of in Situ Oxidation-Generated ortho-Quinone Methides and Aldehydes
2018
Small Molecules Simultaneously Inhibiting p53-Murine Double Minute 2 (MDM2) Interaction and Histone Deacetylases (HDACs): Discovery of Novel Multitargeting Antitumor Agents
2018
Analyte Regeneration Fluorescent Probes for Formaldehyde Enabled by Regiospecific Formaldehyde-Induced Intramolecularity
2018
Recent developments in multimodality fluorescence imaging probes
2018
Discovery of novel indoleamine 2, 3-dioxygenase 1 (IDO1) and histone deacetylase (hdac) dual inhibitors
2018
α-Functionalization of 2-Vinylpyridines via a Chiral Phosphine Catalyzed Enantioselective Cross Rauhut-Currier Reaction
2018
A novel PDE9 inhibitor WYQ-C36D ameliorates corticosterone-induced neurotoxicity and depression-like behaviors by cGMP-CREB-related signaling
2018
Catalytic Cascade Access to Biaryl-2-Methyl Acetates from Pyruvate O-Arylmethyl Ketoximes via the Palladium-Catalyzed C(sp2)-H Bond Arylation and C-O Bond Solvolysis
2018
A pinacol boronate caged NIAD-4 derivative as a near-infrared fluorescent probe for fast and selective detection of hypochlorous acid
2018
Pd-Catalyzed Debenzylation and Deallylation of Ethers and Esters with Sodium Hydride
2018
Alkenylazaarenes as Dipolarophiles in 1,3-Dipolar Cycloaddition of Nitrones: Regioselectivity-Switchable and Highly Diastereoselective Synthesis of Multisubstituted Isoxazolidines
2018
A general asymmetric route to enantio-enriched isoflavanes via an organocatalytic annulation of o-quinone methides and aldehydes
2018
Catalytic Cascade Access to Biaryl‐2‐Methyl Acetates from Pyruvate O‐Arylmethyl Ketoximes via the Palladium‐Catalyzed C(sp2)H Bond Arylation and C−O …
2018
Direct Access of the Chiral Quinolinyl Core of Cinchona Alkaloids via a Brønsted Acid and Chiral Amine Co-catalyzed Chemo- and Enantioselective α-Alkylation of Quinolinylmethanols with Enals
2018
Discovery of Novel Indoleamine 2,3-Dioxygenase 1 (IDO1) and Histone Deacetylase (HDAC) Dual Inhibitors
2018
Direct Access of the Chiral Quinolinyl Core of Cinchona Alkaloids via a Brønsted Acid and Chiral Amine Co-catalyzed Chemo-and Enantioselective α-Alkylation of …
2018
Synthesis of 2-Quinolinones via a Hypervalent Iodine (III)-Mediated Intramolecular Decarboxylative Heck-Type Reaction at Room Temperature
2018
Alkenylazaarenes as dipolarophiles in 1, 3-dipolar cycloaddition of nitrones: regioselectivity-switchable and highly diastereoselective synthesis of multisubstituted isoxazolidines
2018
Small-Molecule Inhibitors for the β-Catenin/T Cell Factor Protein-Protein Interaction
2018
Synthesis of Aldehydes by Organocatalytic Formylation Reactions of Boronic Acids with Glyoxylic Acid
2017
Engineering Iron Responses in Mammalian Cells by Signal-Induced Protein Proximity
2017
A dynamic kinetic asymmetric transfer hydrogenation–cyclization tandem reaction: an easy access to chiral 3, 4-dihydro-2 H-pyran-carbonitriles
2017
Co(OAc)2-Catalyzed Trifluoromethylation and C(3)-Selective Arylation of 2-(Propargylamino)pyridines via a 6-Endo-Dig Cyclization
2017
Iron‐Catalyzed Anti‐Markovnikov Hydroamination of Vinylpyridines
2017
Asymmetric synthesis of isoquinolinonaphthyridines catalyzed by a chiral Brønsted acid
2017
Lewis Acid‐Catalyzed C (sp3)–C (sp3) Bond Forming Cyclization Reactions for the Synthesis of Tetrahydroprotoberberine Derivatives
2017
Visible‐Light‐Promoted Nickel‐and Organic‐Dye‐Cocatalyzed Formylation Reaction of Aryl Halides and Triflates and Vinyl Bromides with Diethoxyacetic Acid as a Formyl Equivalent
2017
Direct Cα-heteroarylation of structurally diverse ethers via a mild N-hydroxysuccinimide mediated cross-dehydrogenative coupling reaction
2017
Palladium‐Catalyzed Divergent Regioselective Homocoupling and Hydroxylation of 3‐Arylbenzo [d] isoxazoles
2017
Orchestration of dual cyclization processes and dual quenching mechanisms for enhanced selectivity and drastic fluorescence turn-on detection of cysteine
2017
An Unconventional Redox Cross Claisen Condensation–Aromatization of 4-Hydroxyprolines with Ketones
2017
Chemo-and regioselective organo-photoredox catalyzed hydroformylation of styrenes via a radical pathway
2017
Synthesis of Z-alkenes via visible light promoted photocatalytic E→ Z isomerization under metal-free conditions
2017
Discovery of IDO1 and DNA dual targeting antitumor agents
2017
Synthesis of Indolizines via Reaction of 2-Substitued Azaarenes with Enals by an Amine-NHC Relay Catalysis
2017
Organocatalytic asymmetric addition of alcohols to cyclic trifluoromethyl ketimines: highly enantioselective synthesis of chiral N, O-ketals
2016
Rational Design of an Ultrasensitive and Highly Selective Chemodosimeter by a Dual Quenching Mechanism for Cysteine Based on a Facile Michael‐Transcyclization Cascade Reaction
2016
Enantioselective synthesis of diarylcyclopropanecarboaldehydes by organocatalysis
2016
Organocatalytic annulation of aldehydes and o-quinone methides: A facile access to dihydrocoumarins
2016
Practical Pd (TFA) 2-Catalyzed Aerobic [4+ 1] Annulation for the Synthesis of Pyrroles via “One-Pot” Cascade Reactions
2016
Facile construction of pyrrolo [1, 2-b] isoquinolin-10 (5 H)-ones via a redox-amination–aromatization–Friedel–Crafts acylation cascade reaction and discovery of novel …
2016
Aniline‐Promoted Cyclization–Replacement Cascade Reactions of 2‐Hydroxycinnamaldehydes with Various Carbonic Nucleophiles through In Situ Formed N, O‐Acetals
2016
A Metal‐free Approach to 3‐Aryl‐3‐hydroxy‐2‐oxindoles by Treatment of 3‐Acyloxy‐2‐oxindoles with Diaryliodonium Salts
2016
Enantioselective organocatalytic Michael addition of isorhodanines to α, β-unsaturated aldehydes
2016
Dynamic kinetic resolution of biaryl lactones via a chiral bifunctional amine thiourea-catalyzed highly atropo-enantioselective transesterification
2016
A mild and selective protecting and reversed modification of thiols
2016
Ligand-free Cu-catalyzed [3+ 2] cyclization for the synthesis of pyrrolo [1, 2-a] quinolines with ambient air as a terminal oxidant
2016
Synthesis of Tryptanthrins by Organocatalytic and Substrate Co-catalyzed Photochemical Condensation of Indoles and Anthranilic Acids with Visible Light and O2
2016
Highly Regio- and Stereoselective Synthesis of Z and E Enol Esters by an Amine-Catalyzed Conjugate Addition–Rearrangement Reaction of Ynals with …
2016
A Multifaceted Directing Group Switching Ynones as Michael Donors in Chemo-, Enantio-, and γ-Selective 1, 4-Conjugate Additions with Nitroolefins
2016
Reaction-based “off–on” fluorescent probe enabling detection of endogenous labile Fe2+ and imaging of Zn2+-induced Fe2+ flux in living cells and elevated Fe2+ in ischemic stroke
2016
Facile Installation of 2‐Reverse Prenyl Functionality into Indoles by a Tandem N‐Alkylation–Aza‐Cope Rearrangement Reaction and Its Application in Synthesis
2016
Synergistic chiral iminium and palladium catalysis: Highly regio-and enantioselective [3+ 2] annulation reaction of 2-vinylcyclopropanes with enals
2016
Stereoselective organocatalytic oxidation of alcohols to enals: a homologation method to prepare polyenes
2016
Enzymatic cleavage and subsequent facile intramolecular transcyclization for in situ fluorescence detection of γ-glutamyltranspetidase activities
2016
β-cyclodextrin-based inclusion complexation bridged biodegradable self-assembly macromolecular micelle for the delivery of paclitaxel
2016
A donor–acceptor triptycene–coumarin hybrid dye featuring a charge separated excited state and AIE properties
2016
New small-molecule drug design strategies for fighting resistant influenza A
2015
Organocatalytic Aerobic Oxidation of Benzylic sp3 C–H Bonds of Ethers and Alkylarenes Promoted by a Recyclable TEMPO Catalyst
2015
State-of-the-art strategies for targeting protein–protein interactions by small-molecule inhibitors
2015
Correction: State-of-the-art strategies for targeting protein–protein interactions by small-molecule inhibitors
2015
Asymmetric synthesis of syn-propargylamines and unsaturated β-amino acids under Brønsted base catalysis
2015
Cross-linked supramolecular polymer metallogels constructed via a self-sorting strategy and their multiple stimulus-response behaviors
2015
Divergent Cascade Construction of Skeletally Diverse “Privileged” Pyrazole‐Derived Molecular Architectures
2015
Amine‐Catalyzed Highly Regioselective and Stereoselective C(sp2)–C(sp2) Cross‐Coupling of Naphthols with trans‐α,β‐Unsaturated Aldehydes
2015
Phosphine-catalyzed Aza-MBH reactions of vinylpyridines: Efficient and rapid access to 2, 3, 5-triarylsubstituted 3-pyrrolines
2015
Construction of an all-carbon quaternary stereocenter by organocatalytic enantioselective α-functionalization of α-substituted β-ketocarbonyls with electron deficient vinylarenes
2015
Divergent Synthesis of Imidazoles and Quinazolines via Pd(OAc)2-Catalyzed Annulation of N-Allylamidines
2015
State-of-the-art strategies for targeting protein-protein interactions by small-molecule inhibitors (vol 44, pg 8238, 2015)
2015
Near-infrared fluorescent probes for imaging of amyloid plaques in Alzheimer׳ s disease
2015
An Efficient Method for the Production of Terminal Alkynes from 1, 1‐Dibromo‐1‐alkenes and its Application in the Total Synthesis of Natural Product Dihydroxerulin
2015
Fluorescent theranostic agents for Hg 2+ detection and detoxification treatment
2015
FeCl3-catalyzed selective acylation of amines with 1, 3-diketones via C–C bond cleavage
2015
Organocatalytic Enantioselective Direct Additions of Aldehydes to 4-Vinylpyridines and Electron-Deficient Vinylarenes and Their Synthetic Applications
2015
Organocatalytic enantioselective Michael addition of cyclic hemiacetals to nitroolefins: A facile access to chiral substituted 5-and 6-membered cyclic ethers
2015
Photo-triggered fluorescent theranostic prodrugs as DNA alkylating agents for mechlorethamine release and spatiotemporal monitoring
2015
Constructing de Novo H2O2 Signaling via Induced Protein Proximity
2015
A Quinine-Squaramide Catalyzed Enantioselective Aza-Friedel–Crafts Reaction of Cyclic Trifluoromethyl Ketimines with Naphthols and Electron-Rich Phenols
2015
Construction of Chiral Bridged Tricyclic Benzopyrans: Enantioselective Catalytic Diels–Alder Reaction and a One‐Pot Reduction/Acid‐Catalyzed Stereoselective Cyclization
2014
One-pot synthesis of 2-substituted benzo [b] furans via Pd–tetraphosphine catalyzed coupling of 2-halophenols with alkynes
2014
Facile Assembly of Chiral Tetrahydrothiopyrans Containing Four Consecutive Stereocenters via an Organocatalytic Enantioselective Michael–Michael Cascade
2014
Enantioselective Construction of Functionalized Cyclopentanes by a Relay Ring-Closing Metathesis and Chiral Amine (Thio) urea-Promoted Michael Addition
2014
Cover Picture: Synthesis of γ‐Oxo‐α,β‐dehydro‐α‐amino Acids from N–tert‐Butyloxycarbonyl‐α‐Imino Esters and Carbonylmethyl 2‐Pyridinylsulfones via an …
2014
PEGylated nickel carbide nanocrystals as efficient near-infrared laser induced photothermal therapy for treatment of cancer cells in vivo
2014
Hollow zeolitic imidazolate framework nanospheres as highly efficient cooperative catalysts for [3+ 3] cycloaddition reactions
2014
Catalytic Asymmetric α‐Hydroxyamination of Carbonyls with N‐Hydroxycarbamates Becomes Greener
2014
Iron/iron oxide core/shell nanoparticles for magnetic targeting MRI and near-infrared photothermal therapy
2014
Highly active, durable and recyclable ordered mesoporous magnetic organometallic catalysts for promoting organic reactions in water
2014
Organocatalytic Enantioselective Friedel–Crafts Reaction of 1‐Naphthols with Isatins and an Unexpected Spontaneous Dehydration Process
2014
Synthesis of γ‐Oxo‐α,β‐dehydro‐α‐amino Acids from N–tert‐Butyloxycarbonyl‐α‐Imino Esters and Carbonylmethyl 2‐Pyridinylsulfones via an Mannich …
2014
4.02 Nucleophilic Addition-Electrophilic Coupling with a Carbanion Intermediate
2014
Water–Medium Organic Reactions Catalyzed by Active and Reusable Pd/Y Heterobimetal–Organic Framework
2013
‘One-pot’synthesis of 4-substituted 1, 5-diaryl-1H-pyrazole-3-carboxylates via lithium tert-butoxide-mediated sterically hindered Claisen condensation and Knorr reaction
2013
Synthesis of Benzoxazoles via an Amine-Catalyzed [4+ 1] Annulation
2013
Quinine-thiourea catalyzed enantioselective hydrophosphonylation of trifluoromethyl 2 (1 H)-quinazolinones
2013
Organocatalytic enantioselective Strecker reaction of cyclic trifluoromethyl-ketoimines
2013
A strategy enabling enantioselective direct conjugate addition of inert aryl methane nucleophiles to enals with a chiral amine catalyst under mild conditions
2013
Inside Back Cover: Imidazolium‐Based Organic–Inorganic Hybrid Silica as a Functional Platform Dramatically Boosts Chiral Organometallics Performance in Asymmetric Catalysis …
2013
C C Bond Formation by Michael Reaction
2013
A novel lactoferrin-modified β-cyclodextrin nanocarrier for brain-targeting drug delivery
2013
A FRET-based ratiometric fluorescent and colorimetric probe for the facile detection of organophosphonate nerve agent mimic DCP
2013
AMINE‐CATALYZED CASCADE REACTIONS
2013
Facile construction of structurally diverse thiazolidinedione-derived compounds via divergent stereoselective cascade organocatalysis and their biological exploratory studies
2013
Formation of Dihydronaphthalenes via Organocatalytic Enatioselective Michael–Aldol Cascade Reactions with Arylalkanes
2013
Chitosan-graft-β-cyclodextrin nanoparticles as a carrier for controlled drug release
2013
Catalytic cascade reactions
2013
Highly enantioselective conjugate addition of nitroalkanes to enones catalyzed by cinchona alkaloid derived primary amine
2013
Asymmetric Synthesis of Chiral Dihydrothiopyrans via an Organocatalytic Enantioselective Formal Thio [3+ 3] Cycloaddition Reaction with Binucleophilic Bisketone Thioethers
2013
Efficient synthesis of highly substituted pyrroles through a Pd (OCOCF 3) 2-catalyzed cascade reaction of 2-alkenal-1, 3-dicarbonyl compounds with primary amines
2013
Imidazolium‐Based Organic–Inorganic Hybrid Silica as a Functional Platform Dramatically Boosts Chiral Organometallics Performance in Asymmetric Catalysis
2013
Direct oxidative conversion of 3-aryl propionaldehydes to 3-aryl acroleins promoted by SOMO catalysis
2012
Synthesis of Highly Functionalized Chiral 3, 3′-Disubstituted Oxindoles via an Organocatalytic Enantioselective Michael Addition of Nitroalkanes to Indolylidenecyanoacetates
2012
Highly active and reusable organometallic catalysts covalently bonded to an ordered mesoporous polymer
2012
Synthesis of 3-substituted 1, 5-aldehyde esters via an organocatalytic highly enantioselective conjugate addition of new carbonylmethyl 2-pyridinylsulfone to enals
2012
Fluorescent probes for the detection of hydrogen sulfide in biological systems
2012
Total synthesis of polyene natural product dihydroxerulin by mild organocatalyzed dehydrogenation of alcohols
2012
Fluoreszenzsonden zum Nachweis von Schwefelwasserstoff in biologischen Systemen
2012
FeCl 3 promoted highly regioselective [3+ 2] cycloaddition of dimethyl 2-vinyl and aryl cyclopropane-1, 1-dicarboxylates with aryl isothiocyanates
2012
Organocatalytic enantioselective conjugate addition of ketones to isatylidine malononitriles
2012
An Organocatalytic Cascade Approach toward Polysubstituted Quinolines and Chiral 1, 4‐Dihydroquinolines–Unanticipated Effect of N‐Protecting Groups
2012
A fluorescent probe capable of detecting H 2 S at submicromolar concentrations in cells
2012
Rational design of a ratiometric fluorescent probe with a large emission shift for the facile detection of Hg 2+
2012
Targeting the Transposase Domain of the DNA Repair Component Metnase to Enhance ChemotherapyTherapeutically Targeting Transposase Domains
2012
Direct Transformation of Simple Enals to 3, 4‐Disubstituted Benzaldehydes under Mild Reaction Conditions via an Organocatalytic Regio‐and Chemoselective Dimerization Cascade
2012
6.22 C–X Bond Formation: Organocatalytic α-Sulfenylation and α-Selenenylation
2012
Expeditious diastereoselective construction of a thiochroman skeleton via a cinchona alkaloid-derived catalyst
2012
A new facile approach to N-alkylpyrroles from direct redox reaction of 4-hydroxy-l-proline with aldehydes
2012
Chiral Pyrrolidine Sulfonamide Catalyzed Enantioselective Michael Addition of Cyclohexanones to Maleimides
2011
Direct stereoselective α-arylation of unmodified enals using an organocatalytic cross-coupling-like reaction
2011
Catalytic Enantioselective Henry Reactions of Isatins: Application in the Concise Synthesis of (S)‐(−)‐Spirobrassinin
2011
Efficient preparation of trans-α,β-unsaturated aldehydes from saturated aldehydes by oxidative enamine catalysis
2011
Cu (II) catalyzed oxidation-[3+ 2] cycloaddition-aromatization cascade: Efficient synthesis of pyrrolo [2, 1-a] isoquinolines
2011
Real-time analysis of the inside-out regulation of lymphocyte function-associated antigen-1 revealed similarities to and differences from very late antigen-4
2011
Organocatalytic enantioselective β-functionalization of aldehydes by oxidation of enamines and their application in cascade reactions
2011
Organocataslysts and methods of use in chemical synthesis
2011
Bifunctional Cinchona Alkaloid Thiourea Catalyzed Highly Efficient, Enantioselective Aza‐Henry Reaction of Cyclic Trifluoromethyl Ketimines: Synthesis of Anti‐HIV Drug DPC 083
2011
Interplay of Direct Stereocontrol and Dynamic Kinetic Resolution in a Bifunctional Amine Thiourea Catalyzed Highly Enantioselective Cascade Michael–Michael Reaction
2011
Proline derivatives
2011
Organocatalytic Enantioselective Friedel− Crafts Reactions of 1-Naphthols with Aldimines
2011
Water-Medium and Solvent-Free Organic Reactions over a Bifunctional Catalyst with Au Nanoparticles Covalently Bonded to HS/SO3H Functionalized Periodic …
2011
Organocatalyzed Highly Enantioselective and anti‐Selective Construction of γ‐Butenolides through Vinylogous Mukaiyama Aldol Reaction
2010
1, 3-Benzodithiole-1, 1, 3, 3-tetraoxide (BDT) as a versatile methylation reagent in catalytic enantioselective Michael addition reaction with enals
2010
Facile Creation of 3‐Indolyl‐3‐hydroxy‐2‐oxindoles by an Organocatalytic Enantioselective Friedel–Crafts Reaction of Indoles with Isatins
2010
“One-Pot” Access to 4 H-Chromenes with Formation of a Chiral Quaternary Stereogenic Center by a Highly Enantioselective Iminium-allenamine Involved Oxa-Michael− Aldol Cascade
2010
NFATc3 contributes to intermittent hypoxia-induced
2010
Rational design of a highly selective and sensitive fluorescent PET probe for discrimination of thiophenols and aliphatic thiols
2010
Synthesis of Chiral 3-Substituted Phthalides by a Sequential Organocatalytic Enantioselective Aldol-Lactonization Reaction. Three-Step Synthesis of (S)-(−)-3 …
2010
Corrigendum to “Enatioselective organocatalytic synthesis of highly functionalized tetrahydrothiophenes by a Michael-aldol cascade reaction”[Tetrahedron Lett. 50 (2009) 2946–2948]
2010
Iminium–Allenamine Cascade Catalysis: One‐Pot Access to Chiral 4H‐Chromenes by a Highly Enantioselective Michael–Michael Sequence
2010
Corrigendum to “Highly enantioselective Michael-cyclization cascade promoted by synergistic asymmetric aminocatalysis and Lewis acid catalysis”[Tetrahedron Lett. 51 (2010) 1742 …
2010
Highly enantioselective Michael-cyclization cascade promoted by synergistic asymmetric aminocatalysis and Lewis acid catalysis
2010
Isoform-specific prolongation of Kv7 (KCNQ) potassium channel opening mediated by new molecular determinants for drug-channel interactions
2010
Periodic mesoporous organometallic silicas with unary or binary organometals inside the channel walls as active and reusable catalysts in aqueous organic reactions
2010
A Simple Primary Amine Thiourea Catalyzed Highly Enantioselective Conjugate Addition of α, α‐Disubstituted Aldehydes to Maleimides
2010
Organocatalytic Enantioselective Conjugate Additions of Heteroatoms to α, βUnsaturated Carbonyl Compounds
2010
Organocatalytic enantioselective Michael addition reactions of fluoromalonates with α, β-unsaturated aldehydes
2010
Highly enantioselective Michael-cyclization cascade promoted by synergistic asymmetric aminocatalysis and Lewis acid catalysis (vol 51, pg 1742, 2010)
2010
Enantioselective cascade michael-michael reactions and related catalysts
2010
NFATc3 contributes to intermittent hypoxia-induced arterial remodeling in mice
2010
Pd-catalyzed cascade Heck–Saegusa: direct synthesis of enals from aryl iodides and allyl alcohol
2010
Diastereo‐and Enantioselective Organocatalytic Direct Conjugate Addition of γ‐Butenolide to Chalcones
2010
Organocatalytic asymmetric synthesis of chiral fluorinated quaternary carbon containing β-ketoesters
2009
Organocatalytic Enantioselective Cross‐Aldol Reactions of Aldehydes with Isatins: Formation of Two Contiguous Quaternary Centered 3‐Substituted 3‐Hydroxyindol‐2‐ones
2009
Conformational mAb as a tool for integrin ligand discovery
2009
Organocatalytic enantioselective conjugate addition of 2-fluoromalonate to nitroolefins: direct synthesis of chiral fluorinated γ-nitro carboxylic acid derivatives
2009
Enantioselective conjugate addition of N-heterocycles to α, β-unsaturated ketones catalyzed by chiral primary amines
2009
Catalytic enantioselective conjugate addition of fluorobis (phenylsulfonyl) methane to enals: synthesis of chiral monofluoromethyl compounds
2009
A selective and sensitive “turn-on” fluorescent chemodosimeter for Hg2+ in aqueous media via Hg2+ promoted facile desulfurization–lactonization reaction
2009
Direct Oxidation of β‐Aryl Substituted Aldehydes to α, β‐Unsaturated Aldehydes Promoted by an o‐Anisidine–Pd (OAc) 2 Co‐catalyst
2009
Enatioselective organocatalytic synthesis of highly functionalized tetrahydrothiophenes by a Michael-aldol cascade reaction
2009
A Direct Amine‐Palladium Acetate Cocatalyzed Saegusa Oxidation Reaction of Unmodified Aldehydes to α, β‐Unsaturated Aldehydes
2009
Catalytic Asymmetric oxa-Michael− Michael Cascade for Facile Construction of Chiral Chromans via an Aminal Intermediate
2009
An Approach to 3, 6-disubstituted 2, 5-dioxybenzoquinones via two sequential Suzuki Couplings. Three-step synthesis of leucomelone
2009
An enantioselective synthesis of (+)-(S)-[n]-gingerols via the l-proline-catalyzed aldol reaction
2009
Simple cyclohexanediamine-derived primary amine thiourea catalyzed highly enantioselective conjugate addition of nitroalkanes to enones
2009
ORGN 598-Enantioselective organocatalytic tandem Michael-aldol reactions: One-pot synthesis of chiral cyclopentenes
2008
Highly enantio-and diastereoselective organocatalytic cascade aza-Michael–Michael reactions: a direct method for the synthesis of trisubstituted chiral pyrrolidines
2008
Enantioselective Cascade Michael-Aldol Condensation Reaction
2008
Activation of Kv7 (KCNQ) voltage-gated potassium channels by synthetic compounds
2008
Organocatalysis: asymmetric cascade reactions catalysed by chiral secondary amines
2008
Total Synthesis of (+)‐Rutamarin
2008
ORGN 596-Enantioselective organocatalytic tandem Michael-aldol reactions
2008
Plk1-dependent phosphorylation of FoxM1 regulates a transcriptional programme required for mitotic progression
2008
Proline-catalyzed direct inverse electron demand Diels–Alder reactions of ketones with 1, 2, 4, 5-tetrazines
2008
An efficient method for demethylation of aryl methyl ethers
2008
ORGN 597-Organocatalytic enantioselective cyclopropanations between alpha, beta-unsaturated aldehydes and bromomalonates
2008
Endothelin 1 activation of NFATc3 contributes to intermittent hypoxia-induced hypertension in mice
2008
An enantioselective formal synthesis of (+)-(R)-α-lipoic acid by an l-proline-catalyzed aldol reaction
2008
Highly enantioselective aldol reactions catalyzed by a recyclable fluorous (S) pyrrolidine sulfonamide on water
2008
Microwave-assisted three-component Knoevenagel-nucleophilic aromatic substitution reactions
2008
Dynamic Kinetic Resolution in an Asymmetric Michael-Michael Cascade
2008
ORGN 599-Tandem Michael-aldol reactions promoted by hydrogen-bonding mediated catalysis
2008
Selective debenzylation of aromatic benzyl ethers by silica-supported sodium hydrogen sulfate
2008
Inverse Diels-Alder Proline-Catalyzed Route to 1, 2, 4, 5-Tetrazines
2008
Hydrogen‐bond‐mediated asymmetric catalysis
2008
A Highly Stereoselective Hydrogen‐Bond‐Mediated Michael–Michael Cascade Process through Dynamic Kinetic Resolution
2008
Chiral Amine‐Catalyzed Enantioselective Cascade Aza–Ene‐Type Cyclization Reactions
2008
An Organocatalytic Approach to the Construction of Chiral Oxazolidinone Rings and Application in the Synthesis of Antibiotic Linezolid and Its Analogues
2008
A novel bifunctional sulfonamide primary amine‐catalyzed enantioselective conjugate addition of ketones to nitroolefins
2008
(S)-Pyrrolidine sulfonamide catalyzed asymmetric direct aldol reactions of aryl methyl ketones with aryl aldehydes
2008
Organocatalytic enantioselective cascade Michael-alkylation reactions: Synthesis of chiral cyclopropanes and investigation of unexpected organocatalyzed stereoselective ring …
2007
Organo-Catalyzed Synthesis of 1, 2-Dihydroquinolines
2007
Chiral Chromenes via Domino Oxa-Michael-Aldol Reaction
2007
An NBD fluorophore-based sensitive and selective fluorescent probe for zinc ion
2007
Conjugate Addition of Nitroalkanes to Nitroolefins
2007
One-pot approach to chiral chromenes via enantioselective organocatalytic domino oxa-Michael–aldol reaction
2007
Cinchona alkaloid based thiourea promoted enantioselective conjugate addition of N-heterocycles to enones
2007
Enantioselective Organocatalytic Domino Michael-Michael Addition Reactions
2007
Highly enantioselective organocatalytic conjugate addition of nitromethane to α, β‐unsaturated aldehydes: three‐step synthesis of optically active baclofen
2007
Enantioselective organocatalytic double Michael addition reactions
2007
Chiral Amine Thiourea‐Promoted Enantioselective Domino Michael‐Aldol Reactions between 2‐Mercaptobenzaldehydes and Maleimides
2007
A Review of:" Analogue-based Drug Discovery"
2007
A highly selective fluorescent probe for thiophenols
2007
Organocatalytic Domino Michael-Aldol Reaction to Chiral Benzothiopyrans
2007
Cascade Michael− aldol reactions promoted by hydrogen bonding mediated catalysis
2007
Highly Enantio-and Diastereoselective Cascade Double Michael Addition
2007
Organocatalytic Enantioselective Cascade Michael–Aldol Condensation Reactions: Efficient Assembly of Densely Functionalized Chiral Cyclopentenes
2007
Erratum: One-pot approach to chiral chromenes via enantioselective organocatalytic domino oxa-Michael-aldol reaction (Chemical Communication (2007)(507-509
2007
Synthesis of Highly Functionalized Chiral Cyclopentanes by Catalytic Enantio‐and Diastereoselective Double Michael Addition Reactions
2007
Quinine‐catalyzed enantioselective Michael addition of diphenyl phosphite to nitroolefins: synthesis of chiral precursors of α‐substituted β‐aminophosphonates
2007
Chiral Diphenylprolinol TES Ether Promoted Conjugate Addition−Aldol-Dehydration Reactions between α,β-Unsaturated Aldehydes and 2-N-Protected Amino …
2007
Organocatalytic enantioselective conjugate additions to enones
2006
Binaphthyl-based bifunctional organocatalyst-promoted enantioselective Morita-Baylis-Hillman reactions
2006
Highly enantioselective organocatalytic Michael addition reactions of ketones with chalcones
2006
Enantioselective organocatalytic Michael addition reactions between N-heterocycles and nitroolefins
2006
Highly enantioselective aldehyde–nitroolefin Michael addition reactions catalyzed by recyclable fluorous (S) diphenylpyrrolinol silyl ether
2006
Organocatalytic One-Pot Synthesis of Chiral Thiochromenes
2006
ORGN 21-(S)-Pyrrolidine sulfonamide and its recyclable version for promoting enantioselective organic reactions in organic and aqueous media
2006
Organocatalysts and methods of use in chemical synthesis
2006
Enantioselective Michael Addition ofN-Heterocycles to Nitroolefins
2006
Binaphthyl-based bifunctional organocatalyst-promoted enantioselective Michael addition of 1, 3-diketones to nitroolefins
2006
Enantioselective Organocatalytic Tandem Michael− Aldol Reactions: One-Pot Synthesis of Chiral Thiochromenes
2006
ORGN 147-Organocatalytic enantioselective Michael addition of thioacetic to nitroolefins and enones
2006
Organocatalytic asymmetric conjugate addition of thioacetic acid to β-nitrostyrenes
2006
A selective and sensitive chemosensor for Cu2+ based on 8-hydroxyquinoline
2006
Chiral pyrrolidine sulfonamide-promoted direct, highly enantio-and diastereoselective Michael addition of ketones to enones
2006
A concise and enantioselective approach to the total synthesis of (−)-lasubine I
2006
ORGN 148-Enantioselective organocatalytic Michael addition of N-heterocycles to nitroolefins and enones
2006
Efficient, enantioselective organocatalytic synthesis of trichostatin A
2006
Organocatalytic enantioselective Michael addition of thioacetic acid to enones
2006
A recyclable fluorous (S)-pyrrolidine sulfonamide promoted direct, highly enantioselective Michael addition of ketones and aldehydes to nitroolefins in water
2006
Organocatalytic, enantioselective conjugate addition of nitroalkanes to nitroolefins
2006
Enantio‐and diastereoselective Michael addition reactions of unmodified aldehydes and ketones with nitroolefins catalyzed by a pyrrolidine sulfonamide
2006
Organocatalytic asymmetric Michael addition of 2, 4-pentandione to nitroolefins
2005
Enantioselective Organocatalytic Mukaiyama− Michael Addition of Silyl Enol Ethers to α, β-Unsaturated Aldehydes
2005
Catalysis of highly stereoselective Mannich-type reactions of aldehydes and ketones with alpha-imino esters by a pyrrolidine sulfonamide: Synthesis of unnatural alpha-amino acids.
2005
A novel pyrrolidine imide catalyzed direct formation of α, β-unsaturated ketones from unmodified ketones and aldehydes
2005
Chiral binaphthyl-derived amine-thiourea organocatalyst-promoted asymmetric Morita− Baylis− Hillman reaction
2005
Direct, Facile Aldehyde and Ketone α-Selenenylation Reactions Promoted by l-Prolinamide and Pyrrolidine Sulfonamide Organocatalysts
2005
Direct, pyrrolidine sulfonamide promoted enantioselective aldol reactions of α, α-dialkyl aldehydes: synthesis of quaternary carbon-containing β-hydroxy carbonyl compounds
2005
Simple, efficient organocatalytic alpha-selenenylation and alpha-sulfenylation reactions of aldehdyes and ketones.
2005
Direct, highly enantioselective pyrrolidine sulfonamide catalyzed Michael addition reactions of aldehydes and ketones to nitrostyrenes and applications for formal synthesis of …
2005
Direct, highly enantioselective pyrrolidine sulfonamide catalyzed Michael addition of aldehydes to nitrostyrenes
2005
Direct, organocatalytic α-sulfenylation of aldehydes and ketones
2004
A Simple and Efficient l-Prolinamide-Catalyzed α-Selenenylation Reaction of Aldehydes
2004
An efficient synthesis of the intrinsic fluorescent peptide labels,(S)-and (R)-(6, 7-dimethoxy-4-coumaryl) alanines via asymmetric hydrogenations
2004
Molecularly imprinted polymers as recognition elements in optical sensors
2004
Catalysis of highly stereoselective Mannich-type reactions of ketones with α-imino esters by a pyrrolidine-sulfonamide. Synthesis of unnatural α-amino acids
2004
An amine sulfonamide organocatalyst for promoting direct, highly enantioselective α-aminoxylation reactions of aldehydes and ketones
2004
Stereoselective synthesis of individual isomers of Leu-enkephalin analogues containing substituted β-turn bicyclic dipeptide mimetics
2003
Stereoselective synthesis of novel dipeptide β-turn mimetics targeting melanocortin peptide receptors
2003
Efficient and stereoselective synthesis of novel cis-4-substituted proline analogues
2003
Practical, asymmetric synthesis of aromatic-substituted bulky and hydrophobic tryptophan and phenylalanine derivatives
2002
An efficient synthesis of (2S, 6S)-and meso-diaminopimelic acids via asymmetric hydrogenation
2002
Delivering peptides and peptidomimetics across membrane barriers: A prodrug approach
2002
Design and synthesis of hydrophobic, bulky χ2-constrained phenylalanine and naphthylalanine derivatives
2002
Design and synthesis of novel χ2-constrained phenylalanine, naphthylalanine, and tryptophan analogues and their use in biologically active melanotropin peptides
2002
Stereoselective synthesis of dipeptide β-turn mimetics: 7-benzyl and 8-phenyl substituted azabicyclo [4.3. 0] nonane amino acid esters
2002
Boronic acid-based sensors
2002
Stereoselective Bromination− Suzuki Cross-Coupling of Dehydroamino Acids To Form Novel Reverse-Turn Peptidomimetics: Substituted Unsaturated and Saturated Indolizidinone Amino …
2002
A General Asymmetric Synthesis of syn- and anti-β-Substituted Cysteine and Serine Derivatives
2002
Regioselective and stereoselective nucleophilic ring opening reactions of a phenyl-substituted aziridine: enantioselective synthesis of β-substituted tryptophan, cysteine, and …
2002
Synthesis of RGD analogs as potential vectors for targeted drug delivery
2001
The development of photometric sensors for boronic acids
2001
Diisopropyl 2‐Allyl‐1, 3, 2‐dioxaborolane‐4, 5‐dicarboxylate
2001
Building fluorescent sensors for carbohydrates using template-directed polymerizations
2001
An efficient approach to asymmetric synthesis of dipeptide β-turn mimetics: indolizidinone amino acids
2001
Practical, asymmetric synthesis of aromatic-substituted bulky and hydrophobic tryptophan derivatives
2001
α, α‐Diphenyl‐2‐pyrrolidinemethanol
2001
1‐Methyl‐2‐pyrrolidinone
2001
A coumarin-based prodrug strategy to improve the oral absorption of RGD peptidomimetics
2000
A facilitated cyclic ether formation and its potential application in solid-phase peptide and organic synthesis
2000
J. Am. Coll. Cardio. J. Am. Coll. Cardio. 27, 536-542, 1996
2000
The first fluorescent sensor for boronic and boric acids with sensitivity at sub-micromolar concentrations
2000
Design, synthesis and evaluation of novel coumarin-based prodrugs and fluorescence sensors
2000
Peptide-Based Drug Design: Controlling Transport and Metabolism Peptide-Based Drug Design: Controlling Transport and Metabolism, 1995
1999
Building fluorescent sensors by template polymerization: the preparation of a fluorescent sensor for D-fructose
1999
Building fluorescent sensors by template polymerization: the preparation of a fluorescent sensor for L-tryptophan
1999
Two new improved approaches to the synthesis of coumarin-based prodrugs
1999
Prodrug approaches to the improved delivery of peptide drugs.
1999
Adv. Drug. Deliv. Res. Adv. Drug. Deliv. Res. 4, 171-207, 1991
1999
Prodrug strategies to improve the oral absorption of peptide mimetics.
1999
Synthesis and evaluation of novel coumarin-based esterase-sensitive cyclic prodrugs of peptidomimetic RGD analogs with improved membrane permeability
1999
Cellular Drug Delivery-Coumarinic Acid-Based Cyclic Prodrugs of Opioid Peptides that Exhibit Metabolic Stability to Peptidases and Excellent Cellular Permeability
1999
Coumarinic acid-based cyclic prodrugs of opioid peptides that exhibit metabolic stability to peptidases and excellent cellular permeability
1999
Synthesis of coumarin-based, esterase-sensitive cyclic prodrugs of opioid peptides with enhanced membrane permeability and enzymatic stability
1999
Lipophilicity in Drug Action and Toxicity Lipophilicity in Drug Action and Toxicity, 233-252, 1996
1999
Biooorg. Med. Chem. Biooorg. Med. Chem. 6, 417-426, 1998
1999
Coumarin-based prodrugs. Part 3: Structural effects on the release kinetics of esterase-sensitive prodrugs of amines
1998
Prodrug strategies to enhance the permeation of opioid peptides through the intestinal mucosa
1998
A comparison of the bioconversion rates and the Caco-2 cell permeation characteristics of coumarin-based cyclic prodrugs and methylester-based linear prodrugs of RGD …
1998
Enantioselective polymeric transporters for tryptophan, phenylalanine, and histidine prepared using molecular imprinting techniques
1998
Peptide science: proceedings of the... Japanese Peptide Symposium 1999, 1-4, 2000-03-01
1997
Chemical feasibility studies of a potential coumarin-based prodrug system
1996

Coumarin-based prodrugs 2. Synthesis and bioreversibility studies of an esterase-sensitive cyclic prodrug of dadle, an opioid peptide
1996

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